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N-Desethylsunitinib hydrochloride
CAS No. 1261432-05-6
N-Desethylsunitinib hydrochloride( —— )
Catalog No. M23434 CAS No. 1261432-05-6
N-Desethylsunitinib hydrochloride is a major and pharmacologically active metabolite of sunitinib, which is potent, ATP-competitive VEGFR, PDGFRβ, and KIT inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 272 | In Stock |
|
| 10MG | 408 | In Stock |
|
| 25MG | 672 | In Stock |
|
| 50MG | 945 | In Stock |
|
| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameN-Desethylsunitinib hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionN-Desethylsunitinib hydrochloride is a major and pharmacologically active metabolite of sunitinib, which is potent, ATP-competitive VEGFR, PDGFRβ, and KIT inhibitor.
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DescriptionN-Desethylsunitinib hydrochloride is a major and pharmacologically active metabolite of sunitinib, which is potent, ATP-competitive VEGFR, PDGFRβ, and KIT inhibitor.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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Targetc-Kit
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RecptorKIT|PDGFRβ|VEGFR
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Research Area——
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Indication——
Chemical Information
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CAS Number1261432-05-6
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Formula Weight406.88
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Molecular FormulaC20H24ClFN4O2
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Purity>98% (HPLC)
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SolubilityDMSO:10 mM
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SMILESO=C1C(C2=CC(F)=CC=C2N1)=CC(NC(C)=C3C(NCCNCC)=O)=C3C.Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Determination of Sunitinib and Its Active Metabolite N-Desethylsunitinib in Sweat of a Patient.[J]. Journal of Analytical Toxicology, 2011.
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